Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50010296
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537192(CHEMBL4563167)
Affinity DataIC50: 240nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537183(CHEMBL4575859)
Affinity DataIC50: 300nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537180(CHEMBL4535649)
Affinity DataIC50: 450nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537194(CHEMBL4528706)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(CHEBI:72292 | Bedaquiline | TMC207)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537181(CHEMBL4522192)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537185(CHEMBL4483435)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537184(CHEMBL4514254)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537190(CHEMBL4521403)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537182(CHEMBL4520823)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537186(CHEMBL4564401)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537192(CHEMBL4563167)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537195(CHEMBL4534128)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537196(CHEMBL4541578)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537180(CHEMBL4535649)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537183(CHEMBL4575859)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537193(CHEMBL4558224)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537191(CHEMBL4522585)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537190(CHEMBL4521403)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537189(CHEMBL4515863)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537188(CHEMBL4515667)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50537187(CHEMBL4574868)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(CHEBI:72292 | Bedaquiline | TMC207)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed