Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50007358
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 7nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 7nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 14nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508783(CHEMBL3325515)
Affinity DataIC50: 16nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 18nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 21nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 26nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 28nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 29nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508787(CHEMBL3325519)
Affinity DataIC50: 34nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508781(CHEMBL4577391)
Affinity DataIC50: 36nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508782(CHEMBL3774725)
Affinity DataIC50: 39nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 49nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508784(CHEMBL4543868)
Affinity DataIC50: 50nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 51nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C double mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 52nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C double mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 55nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508789(CHEMBL3775346)
Affinity DataIC50: 60nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508792(CHEMBL4579182)
Affinity DataIC50: 63nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 73nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 74nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM1434(BI-RG-587 | 2-cyclopropyl-7-methyl-2,4,9,15-tetraa...)
Affinity DataIC50: 105nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 107nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 111nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 126nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 126nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 166nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508781(CHEMBL4577391)
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508781(CHEMBL4577391)
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 236nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188C mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 293nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508791(CHEMBL4439382)
Affinity DataIC50: 303nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 377nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508779(CHEMBL4450185)
Affinity DataIC50: 415nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 468nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508776(CHEMBL4470380)
Affinity DataIC50: 494nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 630nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 798nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 894nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C double mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508777(CHEMBL4438953)
Affinity DataIC50: 926nMAssay Description:Inhibition of HIV1 reverse transcriptase V106M mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188H mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508786(CHEMBL4441079)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508788(CHEMBL4519998)
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508778(CHEMBL4450262)
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508780(CHEMBL4520231)
Affinity DataIC50: 3.88E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508790(CHEMBL4584925)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Stellenbosch University

Curated by ChEMBL
LigandPNGBDBM50508785(CHEMBL4459834)
Affinity DataIC50: 4.41E+4nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase in HIV1 infected HEK293T cells harboring luciferase gene assessed as reduction in viral infection ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed