Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50008299
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517725BDBM50517725(CHEMBL4437602)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517705BDBM50517705(CHEMBL4544986)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517709BDBM50517709(CHEMBL4462878)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517708BDBM50517708(CHEMBL4560346)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517723BDBM50517723(CHEMBL4581107)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517701BDBM50517701(CHEMBL4558181)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517721BDBM50517721(CHEMBL4441549)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517717BDBM50517717(CHEMBL4445307)
Affinity DataIC50: 2.28E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517707BDBM50517707(CHEMBL4520361)
Affinity DataIC50: 3.03E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517719BDBM50517719(CHEMBL4438949)
Affinity DataIC50: 3.78E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517724BDBM50517724(CHEMBL4444366)
Affinity DataIC50: 4.05E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517713BDBM50517713(CHEMBL4466425)
Affinity DataIC50: 7.54E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517704BDBM50517704(CHEMBL4461885)
Affinity DataIC50: 8.88E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517722BDBM50517722(CHEMBL4573983)
Affinity DataIC50: 9.04E+4nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517727BDBM50517727(CHEMBL4582564)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517728BDBM50517728(CHEMBL4462868)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517726BDBM50517726(CHEMBL4561047)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517720BDBM50517720(CHEMBL4462239)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517718BDBM50517718(CHEMBL4577330)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517715BDBM50517715(CHEMBL4576788)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517716BDBM50517716(CHEMBL4449144)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517714BDBM50517714(CHEMBL4476299)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517711BDBM50517711(CHEMBL4532010)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517712BDBM50517712(CHEMBL4459954)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517710BDBM50517710(CHEMBL4457561)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517706BDBM50517706(CHEMBL4540354)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517703BDBM50517703(CHEMBL4466866)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50517702BDBM50517702(CHEMBL4550918)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yanbian University College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148911BDBM50148911(3beta-hydroxyurs-12-en-28-oic acid | (3beta)-3-hyd...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIF1alpha transcriptional activity in human Hep3B cells after 24 hrs in hypoxic condition by HRE-dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed