Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 50009773
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532045(CHEMBL4529550)
Affinity DataEC50:  111nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532027(CHEMBL4529103)
Affinity DataEC50:  848nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532035(CHEMBL4451422)
Affinity DataEC50:  2.04E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532049(CHEMBL4567000)
Affinity DataEC50: >221nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532038(CHEMBL4463066)
Affinity DataEC50:  1.46E+4nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532005(CHEMBL4543208)
Affinity DataEC50:  175nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532048(CHEMBL4536665)
Affinity DataEC50:  183nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532046(CHEMBL4453299)
Affinity DataEC50:  348nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532048(CHEMBL4536665)
Affinity DataEC50:  619nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532009(CHEMBL4440217)
Affinity DataEC50: >5.00E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532037(CHEMBL4457178)
Affinity DataEC50:  176nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532047(CHEMBL4464987)
Affinity DataEC50:  1.93E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532046(CHEMBL4453299)
Affinity DataEC50:  65nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532002(CHEMBL4530409)
Affinity DataEC50:  435nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532044(CHEMBL4559853)
Affinity DataEC50: >3.00E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532023(CHEMBL4454445)
Affinity DataEC50:  1.83E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532043(CHEMBL4476625)
Affinity DataEC50: >4.00E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532022(CHEMBL4540099)
Affinity DataEC50: >3.00E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532003(CHEMBL4475272)
Affinity DataEC50:  1.13E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532020(CHEMBL4451814)
Affinity DataEC50:  1.03E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532018(CHEMBL4470260)
Affinity DataEC50:  1.51E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532042(CHEMBL4518000)
Affinity DataEC50:  850nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532017(CHEMBL4529580)
Affinity DataEC50:  448nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532041(CHEMBL4447978)
Affinity DataEC50:  299nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532015(CHEMBL4550753)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532052(CHEMBL4445429)
Affinity DataEC50:  623nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532004(CHEMBL4593085)
Affinity DataEC50:  4.35E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532021(CHEMBL4540010)
Affinity DataEC50:  998nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532019(CHEMBL4458146)
Affinity DataEC50:  412nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532016(CHEMBL4472955)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532013(CHEMBL4549232)
Affinity DataEC50:  392nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532025(CHEMBL4450006)
Affinity DataEC50:  634nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532047(CHEMBL4464987)
Affinity DataEC50:  4.91E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532030(CHEMBL4459994)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532051(CHEMBL4536856)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532052(CHEMBL4445429)
Affinity DataEC50:  1.26E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532045(CHEMBL4529550)
Affinity DataEC50:  408nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532014(CHEMBL4553987)
Affinity DataEC50:  1.34E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532008(CHEMBL4453946)
Affinity DataEC50:  96nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532051(CHEMBL4536856)
Affinity DataEC50: >5.00E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532050(CHEMBL4447709)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532010(CHEMBL4441816)
Affinity DataEC50:  3.02E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532039(CHEMBL4538108)
Affinity DataEC50:  1.22E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532043(CHEMBL4476625)
Affinity DataEC50:  370nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532006(CHEMBL4593343)
Affinity DataEC50: >1.10E+4nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532042(CHEMBL4518000)
Affinity DataEC50:  183nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532041(CHEMBL4447978)
Affinity DataEC50:  117nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532040(CHEMBL4522066)
Affinity DataEC50:  187nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532044(CHEMBL4559853)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532014(CHEMBL4553987)
Affinity DataEC50:  441nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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