Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50010271
TargetFatty acid-binding protein, adipocyte(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50536996(CHEMBL4581404)
Affinity DataKd:  10nMAssay Description:Binding affinity to recombinant FABP4 (unknown origin) expressed in Escherichia coli by sypro orange dye-based TdF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50536998(CHEMBL4568855)
Affinity DataKd:  860nMAssay Description:Binding affinity to recombinant FABP4 (unknown origin) expressed in Escherichia coli by sypro orange dye-based TdF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetFatty acid-binding protein, adipocyte(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50536999(CHEMBL4547281)
Affinity DataKd:  20nMAssay Description:Binding affinity to recombinant FABP4 (unknown origin) expressed in Escherichia coli by sypro orange dye-based TdF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of California

Curated by ChEMBL
LigandPNGBDBM50193130(CHEMBL3908209)
Affinity DataIC50: 42nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50345442(N-(3,5-Difluoro-4-(trifluoromethyl)phenyl)-5-methy...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human DHODH expressed in Escherichia coli by DCIP staining-based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50536997(CHEMBL4557830)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human DHODH expressed in Escherichia coli by DCIP staining-based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50365230(CHEMBL1956285 | US9238653, Table 5, Compound 10 | ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human DHODH expressed in Escherichia coli by DCIP staining-based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM24400(JMC521864 Compund DSM1 | 5-methyl-N-(naphthalen-2-...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DHODH expressed in Escherichia coli by DCIP staining-based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed