Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50007205
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258769(CHEMBL4096928)
Affinity DataIC50: 18nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258826(CHEMBL4067016)
Affinity DataIC50: 22nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258768(CHEMBL4078901)
Affinity DataIC50: 23nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258766(CHEMBL4077975)
Affinity DataIC50: 27nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258738(CHEMBL4070648)
Affinity DataIC50: 32nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50023629(CHEMBL3341861)
Affinity DataIC50: 33nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507339(CHEMBL4462132)
Affinity DataIC50: 35nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507341(CHEMBL4459402)
Affinity DataIC50: 36nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507343(CHEMBL4513876)
Affinity DataIC50: 40nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507340(CHEMBL4584264)
Affinity DataIC50: 41nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507342(CHEMBL4443345)
Affinity DataIC50: 42nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258802(CHEMBL4089126)
Affinity DataIC50: 47nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50023629(CHEMBL3341861)
Affinity DataIC50: 102nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258768(CHEMBL4078901)
Affinity DataIC50: 151nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507341(CHEMBL4459402)
Affinity DataIC50: 164nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258826(CHEMBL4067016)
Affinity DataIC50: 299nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258769(CHEMBL4096928)
Affinity DataIC50: 353nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507342(CHEMBL4443345)
Affinity DataIC50: 372nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258738(CHEMBL4070648)
Affinity DataIC50: 437nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507340(CHEMBL4584264)
Affinity DataIC50: 440nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258766(CHEMBL4077975)
Affinity DataIC50: 452nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507343(CHEMBL4513876)
Affinity DataIC50: 776nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50507339(CHEMBL4462132)
Affinity DataIC50: 1.38E+3nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50258802(CHEMBL4089126)
Affinity DataIC50: 2.65E+3nMAssay Description:Allosteric modulation of CB1 receptor (unknown origin) assessed as inhibition of CP55940-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed