Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50007285
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508160(CHEMBL4571975)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508160(CHEMBL4571975)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at human PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50135780(2-Methyl-2-(4-{3-[1-(4-methyl-benzyl)-5-oxo-4,5-di...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508126(CHEMBL4457564)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508159(CHEMBL4529735)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508137(CHEMBL4437146)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508153(CHEMBL4549922)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508144(CHEMBL4545223)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508159(CHEMBL4529735)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508127(CHEMBL4449687)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508145(CHEMBL4450146)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508147(CHEMBL4530053)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508151(CHEMBL4449183)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508126(CHEMBL4457564)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50013729(CHEMBL3264919)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508143(CHEMBL4443720)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508155(CHEMBL4592038)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508125(CHEMBL4533138)
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508128(CHEMBL4539262)
Affinity DataIC50: 55nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508132(CHEMBL4546054)
Affinity DataIC50: 56nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508141(CHEMBL4447577)
Affinity DataIC50: 61nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508146(CHEMBL4587456)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508146(CHEMBL4587456)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508150(CHEMBL4547480)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508143(CHEMBL4443720)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508158(CHEMBL4474275)
Affinity DataIC50: 83nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508127(CHEMBL4449687)
Affinity DataIC50: 113nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508157(CHEMBL4471562)
Affinity DataIC50: 122nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508128(CHEMBL4539262)
Affinity DataIC50: 124nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508141(CHEMBL4447577)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508132(CHEMBL4546054)
Affinity DataIC50: 131nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508144(CHEMBL4545223)
Affinity DataIC50: 138nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508153(CHEMBL4549922)
Affinity DataIC50: 197nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508154(CHEMBL4582294)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508145(CHEMBL4450146)
Affinity DataIC50: 216nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508157(CHEMBL4471562)
Affinity DataIC50: 225nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508136(CHEMBL4519021)
Affinity DataIC50: 319nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508148(CHEMBL4566732)
Affinity DataIC50: 394nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508158(CHEMBL4474275)
Affinity DataIC50: 420nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508135(CHEMBL4566043)
Affinity DataIC50: 424nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508142(CHEMBL4452945)
Affinity DataIC50: 433nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508125(CHEMBL4533138)
Affinity DataIC50: 438nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508147(CHEMBL4530053)
Affinity DataIC50: 439nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508142(CHEMBL4452945)
Affinity DataIC50: 515nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508155(CHEMBL4592038)
Affinity DataIC50: 569nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508140(CHEMBL4581797)
Affinity DataIC50: 608nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508151(CHEMBL4449183)
Affinity DataIC50: 610nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508135(CHEMBL4566043)
Affinity DataIC50: 667nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508129(CHEMBL4581233)
Affinity DataIC50: 678nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50508138(CHEMBL4451462)
Affinity DataIC50: 725nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
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