Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50009179
TargetP2X purinoceptor 7(Human)
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50525941(CHEMBL4445773)
Affinity DataIC50: 103nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50525940(CHEMBL4454986)
Affinity DataIC50: 230nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50234965(A-740003 | N-(1-{[(Cyanoimino)(5-quinolinylamino)m...)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Fluminense Federal University

Curated by ChEMBL
LigandPNGBDBM50277548(CHEMBL4173394)
Affinity DataIC50: 1.37E+3nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 5 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed