Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50008617
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520855(CHEMBL4449172)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520856(CHEMBL4437809)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520857(CHEMBL4435565)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520858(CHEMBL4538386)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520859(CHEMBL4524433)
Affinity DataEC50:  163nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50329706((2S)-3-{4-[1-ethyl-1-(4-{[(2R)-2-hydroxy-3,3-dimet...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520860(CHEMBL4558352)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50520861(CHEMBL4583069)
Affinity DataEC50:  9.30nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0110nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed