Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50003075
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466618(CHEMBL4280015)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466619(CHEMBL4290656)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466620(CHEMBL4283481)
Affinity DataKd:  800nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466621(CHEMBL4295184)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed