Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50003322
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469540(CHEMBL4294901)
Affinity DataKd:  0.990nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469541(CHEMBL4289837)
Affinity DataKd:  0.450nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469542(CHEMBL4278500)
Affinity DataKd:  0.320nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469540(CHEMBL4294901)
Affinity DataKd:  0.600nMAssay Description:Binding affinity to human V1A receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469547(CHEMBL4278080)
Affinity DataKd:  29nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469546(CHEMBL4286411)
Affinity DataKd:  46nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50024317(Tetragastrin | CHEMBL120632 | 3-{2-[2-Amino-3-(1H-...)
Affinity DataKd:  22nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469544(CHEMBL4281963)
Affinity DataKi:  0.200nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469541(CHEMBL4289837)
Affinity DataKi:  0.400nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50114031(1-[5-Chloro-3-(2-chloro-phenyl)-1-(3,4-dimethoxy-b...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469540(CHEMBL4294901)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469544(CHEMBL4281963)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50114031(1-[5-Chloro-3-(2-chloro-phenyl)-1-(3,4-dimethoxy-b...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469541(CHEMBL4289837)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469542(CHEMBL4278500)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469540(CHEMBL4294901)
Affinity DataKi:  1.70nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469539(CHEMBL562961)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]OH-LVA from human V1A receptor expressed in African green monkey COS7 cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469541(CHEMBL4289837)
Affinity DataKi:  3.80nMAssay Description:Displacement of [Sez6]-HO-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469539(CHEMBL562961)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469546(CHEMBL4286411)
Affinity DataKi:  3.90nMAssay Description:Displacement of non-sulfated CCK-8 from CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469547(CHEMBL4278080)
Affinity DataKi:  7.90nMAssay Description:Displacement of non-sulfated CCK-8 from CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50024317(Tetragastrin | CHEMBL120632 | 3-{2-[2-Amino-3-(1H-...)
Affinity DataKi:  10nMAssay Description:Displacement of non-sulfated CCK-8 from CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469542(CHEMBL4278500)
Affinity DataKi:  13nMAssay Description:Displacement of [Ph-Se-acetyl]-LVA from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469545(CHEMBL4283439)
Affinity DataKi:  304nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469543(CHEMBL4286989)
Affinity DataKi:  1.28E+3nMAssay Description:Displacement of [125I]OH-Phpa-LVA from human V1A receptor expressed in CHO cells after 4 hrs by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50469545(CHEMBL4283439)
Affinity DataKi:  2.95E+3nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed