Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50007161
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506861(CHEMBL4449031)
Affinity DataIC50: 0.410nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506868(CHEMBL4467278)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506872(CHEMBL4438320)
Affinity DataIC50: 9.5nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506870(CHEMBL4536521)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506867(CHEMBL4516396)
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506866(CHEMBL4534388)
Affinity DataIC50: 89nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506869(CHEMBL4482892)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506871(CHEMBL4475716)
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506861(CHEMBL4449031)
Affinity DataIC50: 780nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in human T47D cells after 20 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506865(CHEMBL4562723)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506864(CHEMBL4528635)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506860(CHEMBL4524233)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506868(CHEMBL4467278)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in human T47D cells after 20 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in human T47D cells after 20 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506862(CHEMBL4575732)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506867(CHEMBL4516396)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in human T47D cells after 20 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
European Institute of Chemistry and Biology (Iecb)

Curated by ChEMBL
LigandPNGBDBM50506863(CHEMBL4446696)
Affinity DataIC50: 1.01E+3nMAssay Description:Displacement of [3H]dexamethasone from GR in human IM9 cells after 6 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed