Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50006804
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503445(CHEMBL4445544 | US11274074, Example 1 [Chemical Fo...)
Affinity DataIC50: 21nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503445(CHEMBL4445544 | US11274074, Example 1 [Chemical Fo...)
Affinity DataIC50: 22nMAssay Description:Inhibition of ANO1 (unknown origin) expressed in FRT cells assessed as reduction in ATP-induced chloride current after 20 mins by electrophysiologica...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50: 77nMAssay Description:Inhibition of ANO1 (unknown origin) expressed in FRT cells assessed as reduction in ATP-induced chloride current after 20 mins by electrophysiologica...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50: 97nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503455(CHEMBL4448175 | US11274074, Example 5 [Chemical Fo...)
Affinity DataIC50: 210nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503439(CHEMBL4515829 | US11274074, Example 6 [Chemical Fo...)
Affinity DataIC50: 300nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503453(CHEMBL4577443)
Affinity DataIC50: 890nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503434(CHEMBL4449467 | US11274074, Example 2 [Chemical Fo...)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503431(CHEMBL4471568 | US11274074, Example 3 [Chemical Fo...)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503440(CHEMBL4441034 | US11274074, Example 7 [Chemical Fo...)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503431(CHEMBL4471568 | US11274074, Example 3 [Chemical Fo...)
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503437(CHEMBL4516441 | US11274074, Example 4 [Chemical Fo...)
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503443(CHEMBL4579558 | US11274074, Example 8 [Chemical Fo...)
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503449(CHEMBL4517769 | US11274074, Example 10 [Chemical F...)
Affinity DataIC50: 3.13E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503440(CHEMBL4441034 | US11274074, Example 7 [Chemical Fo...)
Affinity DataIC50: 5.94E+4nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503442(CHEMBL4453660 | US11274074, Example 9 [Chemical Fo...)
Affinity DataIC50: 6.38E+4nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503454(CHEMBL4472630 | US11274074, Comparative Example 9[)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503433(CHEMBL4462374 | US11274074, Comparative Example 19...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503449(CHEMBL4517769 | US11274074, Example 10 [Chemical F...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503451(CHEMBL4463597 | US11274074, Comparative Example 7 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503430(CHEMBL4586921 | US11274074, Comparative Example 8 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503432(CHEMBL4581421 | US11274074, Comparative Example 11...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503438(CHEMBL4466337 | US11274074, Comparative Example 6 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503446(CHEMBL4434782 | US11274074, Comparative Example 5 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503441(CHEMBL4471557)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503444(CHEMBL4450351 | US11274074, Comparative Example 10...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503438(CHEMBL4466337 | US11274074, Comparative Example 6 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503437(CHEMBL4516441 | US11274074, Example 4 [Chemical Fo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503439(CHEMBL4515829 | US11274074, Example 6 [Chemical Fo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503434(CHEMBL4449467 | US11274074, Example 2 [Chemical Fo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503433(CHEMBL4462374 | US11274074, Comparative Example 19...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503436(CHEMBL4567262 | US11274074, Comparative Example 4 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503435(CHEMBL4465797 | US11274074, Comparative Example 2 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503448(CHEMBL4470594 | US11274074, Comparative Example 1 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503452(CHEMBL4459865 | US11274074, Comparative Example 18...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503435(CHEMBL4465797 | US11274074, Comparative Example 2 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503442(CHEMBL4453660 | US11274074, Example 9 [Chemical Fo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503451(CHEMBL4463597 | US11274074, Comparative Example 7 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO2 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503450(CHEMBL4453183 | US11274074, Comparative Example 17...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503441(CHEMBL4471557)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503447(CHEMBL4476352 | US11274074, Comparative Example 3 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503436(CHEMBL4567262 | US11274074, Comparative Example 4 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50503448(CHEMBL4470594 | US11274074, Comparative Example 1 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YFP-fused ANO1 (unknown origin) expressed in FRT cells after 20 mins by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed