Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50007129
TargetTyrosine-protein kinase Mer(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506638(CHEMBL4465517)
Affinity DataKd:  3.50E+3nMAssay Description:Inhibition of human recombinant GST-tagged cytoplasmic MER (578 to 872 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  19nMAssay Description:Inhibition MER (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506638(CHEMBL4465517)
Affinity DataKd:  6.30E+3nMAssay Description:Inhibition of human recombinant His-tagged AXL (473 to end residues) expressed in insect expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor TYRO3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  7.20E+3nMAssay Description:Inhibition of TYRO3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  12nMAssay Description:Inhibition AXL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human AXL using EAIYAAPFAKKK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506648(CHEMBL4445940)
Affinity DataIC50: 0.940nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 3nMAssay Description:Inhibition of human AuroraA using [H-LRRASLG] as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506636(CHEMBL4445646)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human FLT3 using EAIYAAPFAKKK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human SYK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human PLK1 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 11nMAssay Description:Inhibition of human FAK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 25nMAssay Description:Inhibition of human MER using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor TYRO3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506637(CHEMBL4476226)
Affinity DataIC50: 50nMAssay Description:Inhibition of human TYRO3 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506657(CHEMBL4457670)
Affinity DataIC50: 80nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506649(CHEMBL4546231)
Affinity DataIC50: 790nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506634(CHEMBL4441802)
Affinity DataIC50: 890nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506644(CHEMBL4558560)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506647(CHEMBL4473075)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506641(CHEMBL4460249)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506654(CHEMBL4448090)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506653(CHEMBL4475794)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506656(CHEMBL4463698)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506645(CHEMBL4435161)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506652(CHEMBL4543540)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506651(CHEMBL4461185)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506650(CHEMBL4520283)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506646(CHEMBL4444917)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506643(CHEMBL4553517)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506642(CHEMBL4546644)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506640(CHEMBL4553509)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506639(CHEMBL4531245)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506635(CHEMBL4545017)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50506655(CHEMBL4550527)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of N-terminal His-tagged recombinant human AXL (473 to end amino acids) expressed by baculovirus in Sf9 cells using axltide substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed