Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50003013
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 73nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 85nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 484nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 2.16E+3nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 298nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 96nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 194nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 363nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 86nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 439nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 306nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 121nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 937nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 117nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 1.28E+3nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 634nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 189nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 970nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 483nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 106nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 148nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 171nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 192nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 282nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 303nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 315nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 329nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 369nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 571nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 798nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataIC50: 919nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair
