Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50002881
Affinity DataEC50: 14nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 89nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 95nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 123nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 182nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 182nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 229nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 324nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 363nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 550nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 550nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 560nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 570nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 575nMAssay Description:Agonist activity at rat M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye base...More data for this Ligand-Target Pair
Affinity DataEC50: 575nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 575nMAssay Description:Agonist activity at rat M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye base...More data for this Ligand-Target Pair
Affinity DataEC50: 603nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 604nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Positive allosteric modulation of human M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
Affinity DataEC50: 661nMAssay Description:Agonist activity at human M1 receptor expressed in CHO cells assessed as increase in calcium mobilization measured after 2.5 mins by Fluo-4-AM dye ba...More data for this Ligand-Target Pair
Affinity DataEC50: 759nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 759nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 759nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 760nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 760nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair
Affinity DataEC50: 760nMAssay Description:Positive allosteric modulation of rat M1 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretreate...More data for this Ligand-Target Pair

















