Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50002529
TargetG-protein coupled estrogen receptor 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50303803(cid_5322399 | cid_3136849 | CHEMBL569766 | 1-((3aS...)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50459749(CHEMBL4204236)
Affinity DataEC50:  20nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50459750(CHEMBL4204670)
Affinity DataEC50:  480nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled estrogen receptor 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50459751(CHEMBL4212956)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at GPER (unknown origin) expressed in human HL60 cells assessed as increase in cAMP accumulation in presence of IBMX after 15 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed