Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50002525
TargetFree fatty acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM298452(US10125101, Example 2 | (1S,2S)-2-(5-{(R)-7-Fluoro...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR40 expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50459719(CHEMBL4206195)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human GPR40 expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM298470(US10125101, Example 20)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR40 expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM298482(US10125101, Example 32)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human GPR40 expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM298452(US10125101, Example 2 | (1S,2S)-2-(5-{(R)-7-Fluoro...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR40 expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM298477(US10125101, Example 27)
Affinity DataEC50:  148nMAssay Description:Agonist activity at human GPR40 expressed in human 1321N1 cells assessed as IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed