Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50001914
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450199(CHEMBL4173412)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450187(CHEMBL4166357)
Affinity DataIC50: 480nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450200(CHEMBL4161797)
Affinity DataIC50: 480nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450205(CHEMBL4174659)
Affinity DataIC50: 510nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450206(CHEMBL4174266)
Affinity DataIC50: 530nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450203(CHEMBL4162851)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50442124(CHEMBL2441094)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450186(CHEMBL4167449)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450202(CHEMBL4171945)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450189(CHEMBL4167057)
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450204(CHEMBL4159542)
Affinity DataIC50: 3.40E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450201(CHEMBL4165227)
Affinity DataIC50: 4.30E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450183(CHEMBL4165873)
Affinity DataIC50: 5.30E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450185(CHEMBL4169720)
Affinity DataIC50: 5.70E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450192(CHEMBL4173904)
Affinity DataIC50: 6.30E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450182(CHEMBL4159042)
Affinity DataIC50: 7.40E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450184(CHEMBL4168648)
Affinity DataIC50: 7.60E+3nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450194(CHEMBL4162430)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450195(CHEMBL4173107)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450196(CHEMBL4169303)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450197(CHEMBL4161383)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450198(CHEMBL4164795)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450193(CHEMBL4169699)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450191(CHEMBL4171502)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450190(CHEMBL4174938)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50450188(CHEMBL4160251)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at AR in mouse SC3 cells assessed as inhibition of DHT-induced cell proliferation after 3 days by CCK8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed