Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50003130
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467293(CHEMBL4276825)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50429537(CHEMBL2333770)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467292(CHEMBL4287333)
Affinity DataIC50: 620nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467288(CHEMBL4280909)
Affinity DataIC50: 820nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467291(CHEMBL4279409)
Affinity DataIC50: 2.41E+3nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467290(CHEMBL4277104)
Affinity DataIC50: 7.05E+3nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467284(CHEMBL4292253)
Affinity DataIC50: 7.19E+3nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467286(CHEMBL4294630)
Affinity DataIC50: 7.53E+3nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467287(CHEMBL4287760)
Affinity DataIC50: 9.98E+3nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467285(CHEMBL4284352)
Affinity DataIC50: 1.25E+4nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467289(CHEMBL4278771)
Affinity DataIC50: 1.29E+4nMAssay Description:Antagonist activity at P2Y1 (unknown origin) expressed in human 1321N1 cells assessed as induction of calcium stimulation by fluo-4 dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50373326(CHEMBL444278)
Affinity DataKi:  0.780nMAssay Description:Displacement of [3H]2-chloro-N 6- methyl-( N )-methanocarba-2'-deoxyadenosine 3 ' ,5 '-bis-phosphate from human P2Y1 expressed in baculovirus infecte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)