Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50001910
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50450092(CHEMBL4169451)
Affinity DataKd:  0.400nMAssay Description:Displacement of ARC-1504/ARC-1513-5O from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50450093(CHEMBL4166028)
Affinity DataKd:  48nMAssay Description:Displacement of ARC-1504/ARC-1513-5O from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50450094(CHEMBL4162173)
Affinity DataKd:  0.340nMAssay Description:Displacement of ARC-1504/ARC-1513-5O from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50450095(CHEMBL4172847)
Affinity DataKd:  0.850nMAssay Description:Displacement of ARC-1504/ARC-1513-5O from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50450096(CHEMBL4177303)
Affinity DataKd:  0.580nMAssay Description:Displacement of ARC-1504/ARC-1513-5O from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50: 0.5nMAssay Description:Displacement of 5-TAMRA-labeled ARC-1530 from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50156669(4,5,6,7-tetrabromo-1H-benzimidazole | 4,5,6,7-tetr...)
Affinity DataIC50: 170nMAssay Description:Displacement of 5-TAMRA-labeled ARC-1530 from CK2alpha (unknown origin) (1 to 335 residues) after 15 to 60 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed