Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50003335
TargetDNA (cytosine-5)-methyltransferase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470562(CHEMBL1230055)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human DNMT1A using double-stranded hemi-DNA oligonucleotide as substrate measured after 40 mins by [3H]methyl incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetmRNA cap guanine-N7 methyltransferase(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470562(CHEMBL1230055)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His-tagged RNMT (1 to 476 residues) expressed in Escherichia coli BL21 using 5'-GpppAGAACCUG-biotin-TEG-3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed