Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50002863
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463881(CHEMBL4240336)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to fluorescently labeled recombinant human LSD1 expressed in Escherichia coli by MST analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM101271(US8524717, 26)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463891(CHEMBL4248408)
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463881(CHEMBL4240336)
Affinity DataIC50: 410nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463890(CHEMBL4241311)
Affinity DataIC50: 550nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463885(CHEMBL4245069)
Affinity DataIC50: 870nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463887(CHEMBL4240782)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463880(CHEMBL4244605)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463882(CHEMBL4239151)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463879(CHEMBL4238393)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463884(CHEMBL4251434)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463883(CHEMBL4244132)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463886(CHEMBL4237686)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463888(CHEMBL4237521)
Affinity DataIC50: 6.42E+3nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463892(CHEMBL4248955)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463889(CHEMBL4248864)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463881(CHEMBL4240336)
Affinity DataIC50: 7.25E+4nMAssay Description:Inhibition of recombinant full length N-terminal FLAG-tagged human MAO-A expressed in baculovirus infected Sf9 insect cells using flag peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463878(CHEMBL4250459)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of N-terminal truncated recombinant human LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3 (1 to 21 residues) K4m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50463881(CHEMBL4240336)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant full length N-terminal FLAG-tagged human MAO-B expressed in baculovirus infected Sf9 insect cells using flag peptide as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed