Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50002489
LigandPNGBDBM50459208(CHEMBL4214342)
Affinity DataIC50: 1nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459215(CHEMBL4202685)
Affinity DataIC50: 2nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459203(CHEMBL4207036)
Affinity DataIC50: 2nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459219(CHEMBL4207100)
Affinity DataIC50: 5nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459216(CHEMBL4213673)
Affinity DataIC50: 5nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459201(CHEMBL4217421)
Affinity DataIC50: 6nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459203(CHEMBL4207036)
Affinity DataIC50: 6nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459211(CHEMBL4214863)
Affinity DataIC50: 7nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459209(CHEMBL4209948)
Affinity DataIC50: 8nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459212(CHEMBL4207753)
Affinity DataIC50: 8nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50323777(N-(4-Methyl-3-(1-methyl-7-(6-methylpyridin-3-ylami...)
Affinity DataIC50: 8nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459208(CHEMBL4214342)
Affinity DataIC50: 8nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459216(CHEMBL4213673)
Affinity DataIC50: 9nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459198(CHEMBL4212150)
Affinity DataIC50: 10nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459218(CHEMBL4211976)
Affinity DataIC50: 10nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459207(CHEMBL4212663)
Affinity DataIC50: 11nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459215(CHEMBL4202685)
Affinity DataIC50: 13nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459200(CHEMBL4213019)
Affinity DataIC50: 14nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459199(CHEMBL4215916)
Affinity DataIC50: 15nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459221(CHEMBL4216786)
Affinity DataIC50: 16nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459207(CHEMBL4212663)
Affinity DataIC50: 17nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50242740(Type II inhibitor, 14 | CHEMBL459850 | N-(3-(7-Ami...)
Affinity DataIC50: 18nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459213(CHEMBL4212809)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459209(CHEMBL4209948)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459201(CHEMBL4217421)
Affinity DataIC50: 20nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459197(CHEMBL4209082)
Affinity DataIC50: 21nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459200(CHEMBL4213019)
Affinity DataIC50: 21nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459214(CHEMBL4215989)
Affinity DataIC50: 21nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459220(CHEMBL4203337)
Affinity DataIC50: 23nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459198(CHEMBL4212150)
Affinity DataIC50: 24nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50323777(N-(4-Methyl-3-(1-methyl-7-(6-methylpyridin-3-ylami...)
Affinity DataIC50: 25nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459221(CHEMBL4216786)
Affinity DataIC50: 25nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459212(CHEMBL4207753)
Affinity DataIC50: 25nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459217(CHEMBL4218831)
Affinity DataIC50: 26nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459219(CHEMBL4207100)
Affinity DataIC50: 26nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459202(CHEMBL4211880)
Affinity DataIC50: 27nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459211(CHEMBL4214863)
Affinity DataIC50: 28nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50242740(Type II inhibitor, 14 | CHEMBL459850 | N-(3-(7-Ami...)
Affinity DataIC50: 28nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459218(CHEMBL4211976)
Affinity DataIC50: 28nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459214(CHEMBL4215989)
Affinity DataIC50: 33nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459220(CHEMBL4203337)
Affinity DataIC50: 34nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459205(CHEMBL4210482)
Affinity DataIC50: 35nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459222(CHEMBL4213945)
Affinity DataIC50: 36nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50323778(N-(4-Methyl-3-(1-methyl-2-oxo-7-(phenylamino)-1,2-...)
Affinity DataIC50: 37nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459213(CHEMBL4212809)
Affinity DataIC50: 39nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459204(CHEMBL4206139)
Affinity DataIC50: 40nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetActivated CDC42 kinase 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50459206(CHEMBL4205942)
Affinity DataIC50: 40nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459205(CHEMBL4210482)
Affinity DataIC50: 42nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50459217(CHEMBL4218831)
Affinity DataIC50: 45nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50323778(N-(4-Methyl-3-(1-methyl-2-oxo-7-(phenylamino)-1,2-...)
Affinity DataIC50: 47nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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