Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50003103
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467024(CHEMBL4280697)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50316768((Z,Z)-5-[3-Chloro-4-((2S)-2,3-dihydroxy-propoxy)-b...)
Affinity DataIC50: 13nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467023(CHEMBL4287514)
Affinity DataIC50: 100nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467022(CHEMBL4292022)
Affinity DataIC50: 126nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467025(CHEMBL4288608)
Affinity DataIC50: 316nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467021(CHEMBL4284144)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467026(CHEMBL4285254)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50467027(CHEMBL4292445)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of S1PR1 (unknown origin) expressed in CHOK1 cells after 90 mins by beta-arresting recuitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed