Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50002474
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458989(CHEMBL4215436)
Affinity DataEC50:  14nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458990(CHEMBL4207853)
Affinity DataEC50:  18nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458991(CHEMBL4207315)
Affinity DataEC50:  20nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458992(CHEMBL4212205)
Affinity DataEC50:  20nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458993(CHEMBL4210497)
Affinity DataEC50:  18nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458994(CHEMBL4216650)
Affinity DataEC50:  25nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458995(CHEMBL4212929)
Affinity DataEC50:  22nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458996(CHEMBL4208024)
Affinity DataEC50:  18nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458997(CHEMBL4203670)
Affinity DataEC50:  20nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458998(CHEMBL4202966)
Affinity DataEC50:  14nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50458999(CHEMBL4211671)
Affinity DataEC50:  15nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50459000(CHEMBL4208543)
Affinity DataEC50:  17nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed