Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50002473
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458983(CHEMBL4207166)
Affinity DataIC50: 0.360nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458984(CHEMBL4218897)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458981(CHEMBL4206642)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458979(CHEMBL4210086)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458982(CHEMBL4211530)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458975(CHEMBL4211018)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458978(CHEMBL4214478)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458977(CHEMBL4215980)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458976(CHEMBL4202816)
Affinity DataIC50: 4nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458980(CHEMBL4210884)
Affinity DataIC50: 184nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458987(CHEMBL4206000)
Affinity DataIC50: 197nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.204nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.288nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458979(CHEMBL4210086)
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458979(CHEMBL4210086)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458978(CHEMBL4214478)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458976(CHEMBL4202816)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458978(CHEMBL4214478)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458976(CHEMBL4202816)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458975(CHEMBL4211018)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458984(CHEMBL4218897)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458977(CHEMBL4215980)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458977(CHEMBL4215980)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458982(CHEMBL4211530)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458983(CHEMBL4207166)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458987(CHEMBL4206000)
Affinity DataKi:  28nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458983(CHEMBL4207166)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458981(CHEMBL4206642)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458981(CHEMBL4206642)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458982(CHEMBL4211530)
Affinity DataKi:  33nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458980(CHEMBL4210884)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458984(CHEMBL4218897)
Affinity DataKi:  39nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458975(CHEMBL4211018)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458980(CHEMBL4210884)
Affinity DataKi:  54nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458985(CHEMBL4218247)
Affinity DataKi:  59nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458974(CHEMBL4206516)
Affinity DataKi:  186nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458987(CHEMBL4206000)
Affinity DataKi:  295nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458985(CHEMBL4218247)
Affinity DataKi:  331nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458988(CHEMBL4209446)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458988(CHEMBL4209446)
Affinity DataKi:  447nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458974(CHEMBL4206516)
Affinity DataKi:  603nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458986(CHEMBL4214348)
Affinity DataKi:  3.09E+3nMAssay Description:Displacement of [125I]iodomelatonin from human MT1 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50458986(CHEMBL4214348)
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of [125I]iodomelatonin from human MT2 receptor expressed in rat NIH/3T3 cell membranes incubated for 90 mins by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed