Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002833
Target72 kDa type IV collagenase(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463546(CHEMBL4245382)
Affinity DataIC50: 102nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) preincubated for 45 mins followed by Mea-Pro-Leu-Gly-Leu-Dap(Dnp)-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463546(CHEMBL4245382)
Affinity DataIC50: 162nMAssay Description:Inhibition of recombinant human MMP9 (Phe107 to Pro449 residues) expressed in Escherichia coli preincubated for 45 mins followed by Mea-Pro-Leu-Gly-L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463544(CHEMBL4241167)
Affinity DataIC50: 182nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) preincubated for 45 mins followed by Mea-Pro-Leu-Gly-Leu-Dap(Dnp)-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463544(CHEMBL4241167)
Affinity DataIC50: 242nMAssay Description:Inhibition of recombinant human MMP9 (Phe107 to Pro449 residues) expressed in Escherichia coli preincubated for 45 mins followed by Mea-Pro-Leu-Gly-L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50247539(N-((3S,5S)-1-((E)-3-(3,4-dimethoxyphenyl)acryloyl)...)
Affinity DataIC50: 266nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) preincubated for 45 mins followed by Mea-Pro-Leu-Gly-Leu-Dap(Dnp)-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463547(CHEMBL4249544)
Affinity DataIC50: 345nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) preincubated for 45 mins followed by Mea-Pro-Leu-Gly-Leu-Dap(Dnp)-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50247539(N-((3S,5S)-1-((E)-3-(3,4-dimethoxyphenyl)acryloyl)...)
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant human MMP9 (Phe107 to Pro449 residues) expressed in Escherichia coli preincubated for 45 mins followed by Mea-Pro-Leu-Gly-L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463547(CHEMBL4249544)
Affinity DataIC50: 388nMAssay Description:Inhibition of recombinant human MMP9 (Phe107 to Pro449 residues) expressed in Escherichia coli preincubated for 45 mins followed by Mea-Pro-Leu-Gly-L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463545(CHEMBL4238489)
Affinity DataIC50: 414nMAssay Description:Inhibition of recombinant human MMP2 catalytic domain (Tyr110 to Asp452 residues) preincubated for 45 mins followed by Mea-Pro-Leu-Gly-Leu-Dap(Dnp)-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Weifang Medical University

Curated by ChEMBL
LigandPNGBDBM50463545(CHEMBL4238489)
Affinity DataIC50: 524nMAssay Description:Inhibition of recombinant human MMP9 (Phe107 to Pro449 residues) expressed in Escherichia coli preincubated for 45 mins followed by Mea-Pro-Leu-Gly-L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed