Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50002812
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463350(CHEMBL4243580)
Affinity DataEC50: >5.00E+3nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463351(CHEMBL4240212)
Affinity DataEC50:  12nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463352(CHEMBL4238053)
Affinity DataEC50:  4nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463353(CHEMBL4248974)
Affinity DataEC50:  18nMAssay Description:Activation of p53 in human MCF7 cell lysates assessed as increase in total p53 protein level by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463354(CHEMBL4246320)
Affinity DataEC50:  4nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463355(CHEMBL4240977)
Affinity DataEC50:  152nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463353(CHEMBL4248974)
Affinity DataEC50:  2nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463356(CHEMBL4240141)
Affinity DataEC50:  74nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463357(CHEMBL4243377)
Affinity DataEC50:  158nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463358(CHEMBL4244338)
Affinity DataEC50:  65nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCellular tumor antigen p53(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50463359(CHEMBL4243509)
Affinity DataEC50:  9nMAssay Description:Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed