Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50007124
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506597(CHEMBL4576477)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50175811(N-(4-{[4-(1H-benzoimidazol-2-yl)phenylamino]methyl...)
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50466645(CHEMBL4294823)
Affinity DataIC50: 640nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506608(CHEMBL4564079)
Affinity DataIC50: 820nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506607(CHEMBL4446276)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506598(CHEMBL4455617)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506606(CHEMBL4467480)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506599(CHEMBL4569106)
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506603(CHEMBL4546209)
Affinity DataIC50: 2.56E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506595(CHEMBL4558464)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50466625(CHEMBL4284206)
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506596(CHEMBL4552505)
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506600(CHEMBL4517524)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506604(CHEMBL4551505)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506605(CHEMBL4559163)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506602(CHEMBL4456621)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHeparanase(Human)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50506601(CHEMBL4574859)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant HPSE GS3 (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 based colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed