Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50002776
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462847(CHEMBL4246334)
Affinity DataEC50:  2.40E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462859(CHEMBL4239572)
Affinity DataEC50:  5.04E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462856(CHEMBL4246529)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462855(CHEMBL4242595)
Affinity DataEC50:  463nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462858(CHEMBL4239630)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462848(CHEMBL4238809)
Affinity DataEC50:  2.44E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462851(CHEMBL4240607)
Affinity DataEC50:  6.88E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462859(CHEMBL4239572)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462857(CHEMBL4243863)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as increase in calcium flux measured every 2 secs for 90 secs by Calcium-3 dye bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462854(CHEMBL4246850)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human GPR120More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462854(CHEMBL4246850)
Affinity DataEC50:  1.47E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462858(CHEMBL4239630)
Affinity DataEC50:  874nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462857(CHEMBL4243863)
Affinity DataEC50:  347nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462852(CHEMBL4250132)
Affinity DataEC50:  638nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462856(CHEMBL4246529)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462846(CHEMBL4246396)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462855(CHEMBL4242595)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462854(CHEMBL4246850)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462850(CHEMBL4248845)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462853(CHEMBL4250196)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462853(CHEMBL4250196)
Affinity DataEC50:  2.94E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462852(CHEMBL4250132)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human GPR120 expressed in baculovirus infected sf9 cells assessed as increase in calcium flux measured every 1 sec for 60 secs by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462849(CHEMBL4250664)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462851(CHEMBL4240607)
Affinity DataEC50:  186nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462850(CHEMBL4248845)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462849(CHEMBL4250664)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462846(CHEMBL4246396)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462848(CHEMBL4238809)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50462847(CHEMBL4246334)
Affinity DataEC50:  3.48E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed