Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50001485
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281369(CHEMBL4162750)
Affinity DataIC50: 600nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281371(CHEMBL4171368)
Affinity DataIC50: 600nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281371(CHEMBL4171368)
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281374(CHEMBL4160103)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281371(CHEMBL4171368)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281377(CHEMBL4170169)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281375(CHEMBL4166919)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281384(CHEMBL4170320)
Affinity DataIC50: 4.47E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281383(CHEMBL4163469)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281380(CHEMBL4174506)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281378(CHEMBL4175502)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281376(CHEMBL4174813)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281371(CHEMBL4171368)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281381(CHEMBL4159383)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281386(CHEMBL4176397)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281372(CHEMBL4162255)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281373(CHEMBL4176810)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281382(CHEMBL4168533)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281385(CHEMBL4173454)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281370(CHEMBL4168028)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281387(CHEMBL4166593)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281371(CHEMBL4171368)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281379(CHEMBL4166194)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281376(CHEMBL4174813)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281376(CHEMBL4174813)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases-Diagnostics

Curated by ChEMBL
LigandPNGBDBM50281376(CHEMBL4174813)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of radioligand binding to human ERG expressed in HEK293 cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed