Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50001302
LigandPNGBDBM200324(US9227956, 9)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM200332(US9227956, 16)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM200332(US9227956, 16)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50275434(CHEMBL4127458)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM200332(US9227956, 16)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50275434(CHEMBL4127458)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM200332(US9227956, 16)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50275434(CHEMBL4127458)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM200332(US9227956, 16)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50275434(CHEMBL4127458)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275433(CHEMBL4127311)
Affinity DataIC50: 4.32E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275434(CHEMBL4127458)
Affinity DataIC50: 5.98E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275437(CHEMBL4129620)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM200318(US9227956, 3)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275430(CHEMBL4130157)
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM200324(US9227956, 9)
Affinity DataKi:  5.90E+3nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275486(CHEMBL4128560)
Affinity DataKi:  1.27E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275436(CHEMBL4128250)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275433(CHEMBL4127311)
Affinity DataKi:  1.41E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275485(CHEMBL4126894)
Affinity DataKi:  1.58E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275484(CHEMBL4128388)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM200332(US9227956, 16)
Affinity DataKi:  1.81E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM200320(US9227956, 5)
Affinity DataKi:  2.88E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275487(CHEMBL4126496)
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275434(CHEMBL4127458)
Affinity DataKi:  3.82E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275435(CHEMBL4126072)
Affinity DataKi:  3.84E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50275431(CHEMBL4127016)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of dofetilide binding to human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details Article
PubMed