Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50001297
TargetOxoeicosanoid receptor 1(Human)
Hospital Del Mar Medical Research Institute (Imim)

Curated by ChEMBL
LigandPNGBDBM50027524(5-Oxo-icosa-6,8,11,14-tetraenoic acid methyl ester...)
Affinity DataEC50:  1.54E+3nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetOxoeicosanoid receptor 1(Human)
Hospital Del Mar Medical Research Institute (Imim)

Curated by ChEMBL
LigandPNGBDBM50024458(ETE-5-Oxo | CHEMBL18028 | 5-oxo-ETE)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetOxoeicosanoid receptor 1(Human)
Hospital Del Mar Medical Research Institute (Imim)

Curated by ChEMBL
LigandPNGBDBM50275215(CHEMBL4128585)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetOxoeicosanoid receptor 1(Human)
Hospital Del Mar Medical Research Institute (Imim)

Curated by ChEMBL
LigandPNGBDBM50275216(CHEMBL4130040)
Affinity DataEC50:  2.08E+3nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetOxoeicosanoid receptor 1(Human)
Hospital Del Mar Medical Research Institute (Imim)

Curated by ChEMBL
LigandPNGBDBM50275217(CHEMBL4127146)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed
TargetOxoeicosanoid receptor 1(Human)
Hospital Del Mar Medical Research Institute (Imim)

Curated by ChEMBL
LigandPNGBDBM50275229(CHEMBL4128214)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2020
Entry Details Article
PubMed