Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50001280
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataKd:  10nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) expressed in Escherichia coli BL21-Cod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataKd:  1.5nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human HSP90alpha expressed in Escherichia coli by fluorescence anisotropy methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataIC50: 21nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human HSP90alpha expressed in Escherichia coli by fluorescence anisotropy methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50031735(CHEMBL3360305)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50361703(CHEMBL1941052)
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274536(CHEMBL3900791)
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274534(CHEMBL4128056)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274533(CHEMBL4129436)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274525(CHEMBL4127843)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50361701(CHEMBL1941050)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274518(CHEMBL4128206)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2020
Entry Details Article
PubMed