Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50001273
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274497(CHEMBL4127627)
Affinity DataIC50: 39nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274495(CHEMBL4126401)
Affinity DataIC50: 66nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274494(CHEMBL4128878)
Affinity DataIC50: 70nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274500(CHEMBL4126831)
Affinity DataIC50: 74nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274517(CHEMBL4129028)
Affinity DataIC50: 75nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274496(CHEMBL4127785)
Affinity DataIC50: 78nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274499(CHEMBL4130094)
Affinity DataIC50: 90nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274498(CHEMBL4127365)
Affinity DataIC50: 283nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274496(CHEMBL4127785)
Affinity DataIC50: 716nMAssay Description:Inhibition of FITC-GPMQTSpTPKNG-OH binding to Plk2 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274516(CHEMBL4130239)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of FITC-GPMQSpTPLNG-OH binding to Plk1 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274498(CHEMBL4127365)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of FITC-GPMQTSpTPKNG-OH binding to Plk2 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50274497(CHEMBL4127627)
Affinity DataIC50: 2.54E+4nMAssay Description:Inhibition of FITC-GPLATSpTPKNG-OH binding to Plk3 PBD (unknown origin) after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2020
Entry Details Article
PubMed