Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50003242
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468430(CHEMBL4283085)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468427(CHEMBL1812101)
Affinity DataEC50:  162nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468432(CHEMBL4285396)
Affinity DataEC50:  256nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468430(CHEMBL4283085)
Affinity DataEC50:  834nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  80nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468431(CHEMBL408326)
Affinity DataEC50:  1.59E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468428(CHEBI:44612 | CHEMBL1234965)
Affinity DataEC50:  30nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468429(CHEMBL4279608)
Affinity DataEC50:  815nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468424(CHEMBL4287516)
Affinity DataEC50:  3.46E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468429(CHEMBL4279608)
Affinity DataEC50:  906nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468424(CHEMBL4287516)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468425(CHEBI:56080 | CHEMBL208383)
Affinity DataEC50:  1.38E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468428(CHEBI:44612 | CHEMBL1234965)
Affinity DataEC50:  3.32E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468427(CHEMBL1812101)
Affinity DataEC50:  359nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468425(CHEBI:56080 | CHEMBL208383)
Affinity DataEC50:  110nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468432(CHEMBL4285396)
Affinity DataIC50: 2.50E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ tr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468426(CHEMBL3235593)
Affinity DataIC50: 2.50E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468426(CHEMBL3235593)
Affinity DataIC50: 2.50E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ tr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed