Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50001262
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274076(CHEMBL1384623)
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274068(CHEMBL1411671)
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274074(CHEMBL4127454)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM42435(MLS000729082 | 4-methylbenzyl 5-amino-2-phenyl-2H-...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM48290(cid_2302856 | SMR000153404 | MLS000566310 | N-(1H-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274071(CHEMBL4128696)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274072(CHEMBL4126042)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274070(CHEMBL4129358)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274073(CHEMBL4126651)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274067(CHEMBL4128108)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274073(CHEMBL4126651)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274076(CHEMBL1384623)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274068(CHEMBL1411671)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM42435(MLS000729082 | 4-methylbenzyl 5-amino-2-phenyl-2H-...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in cell membranes after 60 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274072(CHEMBL4126042)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274071(CHEMBL4128696)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274067(CHEMBL4128108)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in cell membranes after 60 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274074(CHEMBL4127454)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274070(CHEMBL4129358)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM48290(cid_2302856 | SMR000153404 | MLS000566310 | N-(1H-...)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]ZM241385 from A2A receptor in human HeLa cell membranes after 30 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274069(CHEMBL4128848)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from A3 receptor in human HeLa cell membranes after 180 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50274075(CHEMBL1561896)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from A3 receptor in human HeLa cell membranes after 180 mins by beta-scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed