Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50001256
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50426994(CHEMBL2326533)
Affinity DataIC50: 11nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50426994(CHEMBL2326533)
Affinity DataIC50: 28nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274010(CHEMBL4126411)
Affinity DataIC50: 119nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274036(CHEMBL4128478)
Affinity DataIC50: 130nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274036(CHEMBL4128478)
Affinity DataIC50: 130nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50273999(CHEMBL4129702)
Affinity DataIC50: 140nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274011(CHEMBL4125911)
Affinity DataIC50: 150nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274033(CHEMBL4128898)
Affinity DataIC50: 200nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274026(CHEMBL4129220)
Affinity DataIC50: 200nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274034(CHEMBL4128074)
Affinity DataIC50: 210nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274035(CHEMBL4129042)
Affinity DataIC50: 210nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274033(CHEMBL4128898)
Affinity DataIC50: 220nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274034(CHEMBL4128074)
Affinity DataIC50: 250nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274041(CHEMBL4127967)
Affinity DataIC50: 300nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274008(CHEMBL4126693)
Affinity DataIC50: 350nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50273999(CHEMBL4129702)
Affinity DataIC50: 360nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274010(CHEMBL4126411)
Affinity DataIC50: 395nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274011(CHEMBL4125911)
Affinity DataIC50: 400nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274033(CHEMBL4128898)
Affinity DataIC50: 450nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274041(CHEMBL4127967)
Affinity DataIC50: 470nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274009(CHEMBL4130258)
Affinity DataIC50: 700nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50273998(CHEMBL4129319)
Affinity DataIC50: 700nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274033(CHEMBL4128898)
Affinity DataIC50: 950nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274043(CHEMBL4127928)
Affinity DataIC50: 980nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-10(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274026(CHEMBL4129220)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274046(CHEMBL4130108)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50426994(CHEMBL2326533)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274035(CHEMBL4129042)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50426994(CHEMBL2326533)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274036(CHEMBL4128478)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274011(CHEMBL4125911)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274011(CHEMBL4125911)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274036(CHEMBL4128478)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274026(CHEMBL4129220)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274026(CHEMBL4129220)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274010(CHEMBL4126411)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274010(CHEMBL4126411)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50273998(CHEMBL4129319)
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274008(CHEMBL4126693)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274009(CHEMBL4130258)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274043(CHEMBL4127928)
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274046(CHEMBL4130108)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274041(CHEMBL4127967)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274041(CHEMBL4127967)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274034(CHEMBL4128074)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50273999(CHEMBL4129702)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-8(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50273999(CHEMBL4129702)
Affinity DataIC50: 1.37E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of Glasgow

Curated by ChEMBL
LigandPNGBDBM50274034(CHEMBL4128074)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details Article
PubMed