Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50001223
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 220447BDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataIC50: 1nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273481BDBM50273481(CHEMBL4125931)
Affinity DataIC50: 18nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273482BDBM50273482(CHEMBL4127310)
Affinity DataIC50: 100nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399434BDBM50399434(CHEMBL2179387)
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365463BDBM50365463(CHEMBL1232461)
Affinity DataIC50: 630nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273496BDBM50273496(CHEMBL4125924)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032921BDBM50032921(CHEMBL1444120)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273497BDBM50273497(CHEMBL4129632)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273483BDBM50273483(CHEMBL4129169)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032911BDBM50032911(CHEMBL1535485)
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273480BDBM50273480(CHEMBL4126342)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50271103BDBM50271103(CHEMBL4129770)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273493BDBM50273493(CHEMBL4127163)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273495BDBM50273495(CHEMBL4127306)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273484BDBM50273484(CHEMBL4127934)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270480BDBM50270480(CHEMBL4126540)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Bienta/Enamine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273479BDBM50273479(CHEMBL4128551)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged BRD4 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2020
Entry Details Article
PubMed