Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50002709
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)
Affinity DataIC50: 750nMAssay Description:Inhibition of human alpha9/alpha10 G154N mutant nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)
Affinity DataIC50: 750nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (3:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (1:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)
Affinity DataIC50: 3.57E+3nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461913(CHEMBL4225280)
Affinity DataIC50: 8.59E+3nMAssay Description:Inhibition of human alpha9 N154G mutant/alpha10 nACHR (3:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461912(CHEMBL4228263)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (3:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461913(CHEMBL4225280)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human alpha9 N154G mutant/alpha10 nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461913(CHEMBL4225280)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (3:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of human alpha9 N154G mutant/alpha10 nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461912(CHEMBL4228263)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human alpha9 N154G mutant/alpha10 nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461912(CHEMBL4228263)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461912(CHEMBL4228263)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human alpha9 N154G mutant/alpha10 nACHR (3:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461911(CHEMBL4229033)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human alpha9 N154G mutant/alpha10 nACHR (3:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461913(CHEMBL4225280)
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (1:3) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461914(CHEMBL4228783)
Affinity DataIC50: 2.22E+4nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (1:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50461915(CHEMBL4226390)
Affinity DataIC50: 2.49E+5nMAssay Description:Inhibition of human alpha9/alpha10 nACHR (1:1) expressed in Xenopus laevis oocyte assessed as inhibition of ACh induced channel current measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed