Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50001837
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405927BDBM50405927(CHEMBL4177351)
Affinity DataIC50: 77nMAssay Description:Inhibition of BRD4 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50071106BDBM50071106(CHEMBL3410002)
Affinity DataIC50: 140nMAssay Description:Inhibition of BRD4 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399434BDBM50399434(CHEMBL2179387)
Affinity DataIC50: 220nMAssay Description:Inhibition of BRD4 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405923BDBM50405923(CHEMBL4175673)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405924BDBM50405924(CHEMBL4165055)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405925BDBM50405925(CHEMBL4159075)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405926BDBM50405926(CHEMBL4171143)
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238042BDBM50238042(CHEMBL4073350)
Affinity DataIC50: 6.83E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405953BDBM50405953(CHEMBL4167326)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405919BDBM50405919(CHEMBL4163466)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405921BDBM50405921(CHEMBL4170290)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406028BDBM50406028(CHEMBL4170804)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406024BDBM50406024(CHEMBL4174139)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406023BDBM50406023(CHEMBL4165445)
Affinity DataIC50: 2.31E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406027BDBM50406027(CHEMBL4162367)
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405922BDBM50405922(CHEMBL4167407)
Affinity DataIC50: 3.22E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238043BDBM50238043(CHEMBL4100505)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406026BDBM50406026(CHEMBL4169300)
Affinity DataIC50: 4.22E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406025BDBM50406025(CHEMBL4177508)
Affinity DataIC50: 4.73E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406030BDBM50406030(CHEMBL4160166)
Affinity DataIC50: 5.08E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Hebei University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50406022BDBM50406022(CHEMBL4172354)
Affinity DataIC50: 6.92E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed