Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50002752
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM99471(US8497274, 32)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM99471(US8497274, 32)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF V600E mutant (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462458(CHEMBL4237480)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462457(CHEMBL4241641)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462456(CHEMBL4246643)
Affinity DataIC50: 74nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF V600E mutant (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462459(CHEMBL4237730)
Affinity DataIC50: 74nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF V600E mutant (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462456(CHEMBL4246643)
Affinity DataIC50: 86nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462459(CHEMBL4237730)
Affinity DataIC50: 87nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462461(CHEMBL4243806)
Affinity DataIC50: 168nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF V600E mutant (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462460(CHEMBL4239581)
Affinity DataIC50: 352nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF V600E mutant (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462462(CHEMBL4243306)
Affinity DataIC50: 421nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF V600E mutant (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462462(CHEMBL4243306)
Affinity DataIC50: 537nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462461(CHEMBL4243806)
Affinity DataIC50: 616nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50462460(CHEMBL4239581)
Affinity DataIC50: 732nMAssay Description:Inhibition of N-terminal 6x-His-tagged BRAF kinase domain (unknown origin) expressed in baculovirus infected Sf9 insect cells co-expressing mouse p50...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed