Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50001214
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272550(CHEMBL4127584)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272568(CHEMBL4128556)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272566(CHEMBL4127168)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272547(CHEMBL4129772)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272565(CHEMBL4128404)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50142759(N-(4-{(R)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-e...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272556(CHEMBL4125820)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272554(CHEMBL4128423)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272553(CHEMBL4129787)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272549(CHEMBL4125928)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272548(CHEMBL4127436)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272534(CHEMBL4126363)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272535(CHEMBL4129117)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272552(CHEMBL4129651)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272551(CHEMBL4126214)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272548(CHEMBL4127436)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272550(CHEMBL4127584)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272551(CHEMBL4126214)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50142759(N-(4-{(R)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-e...)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272554(CHEMBL4128423)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272565(CHEMBL4128404)
Affinity DataIC50: 96nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272534(CHEMBL4126363)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272553(CHEMBL4129787)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272535(CHEMBL4129117)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272568(CHEMBL4128556)
Affinity DataIC50: 240nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272566(CHEMBL4127168)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272547(CHEMBL4129772)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272549(CHEMBL4125928)
Affinity DataIC50: 680nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272556(CHEMBL4125820)
Affinity DataIC50: 680nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50272552(CHEMBL4129651)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2020
Entry Details Article
PubMed