Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50002354
Affinity DataKd: 8nMAssay Description:Binding affinity to PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to KIT (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
University of The Pacific
Curated by ChEMBL
University of The Pacific
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to PDGFRalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Binding affinity to KIT D816V mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to KIT V559D mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding affinity to KIT V559D/T670I mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Binding affinity to KIT V816H mutant (unknown origin)More data for this Ligand-Target Pair
