Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50002689
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50241203(exenatide | HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGSPPP...)
Affinity DataEC50:  0.00180nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461653(CHEMBL509016)
Affinity DataEC50:  0.00560nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461654(CHEMBL4225369)
Affinity DataEC50:  0.0260nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461655(CHEMBL4227957)
Affinity DataEC50:  0.00930nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461656(CHEMBL4227488)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461657(CHEMBL4229047)
Affinity DataEC50:  0.00610nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461658(CHEMBL4228978)
Affinity DataEC50:  0.0140nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461659(CHEMBL4228144)
Affinity DataEC50:  0.00560nMAssay Description:Agonist activity at recombinant human GLP1 receptor expressed in HEK293 cells assessed as cAMP accumulation by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed