Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50001203
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Amherst College

Curated by ChEMBL
LigandPNGBDBM50272021(CHEMBL4128743)
Affinity DataIC50: 125nMAssay Description:Inhibition of allosterically sensitized His6-tagged human PTP1B catalytic domain P87C/A122C mutant using pNPP as substrate incubated for 90 mins by q...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Amherst College

Curated by ChEMBL
LigandPNGBDBM50272021(CHEMBL4128743)
Affinity DataIC50: 125nMAssay Description:Inhibition of allosterically sensitized His6-tagged human PTP1B catalytic domain P87C/A122C mutant overexpressed in Escherichia coli crude cell lysat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Human)
Amherst College

Curated by ChEMBL
LigandPNGBDBM50272020(CHEMBL454668 | CHEBI:52107)
Affinity DataIC50: 125nMAssay Description:Inhibition of allosterically sensitized mutant form of His6-tagged human HePTP catalytic domain using pNPP as substrate incubated for 90 mins by quen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Human)
Amherst College

Curated by ChEMBL
LigandPNGBDBM50272020(CHEMBL454668 | CHEBI:52107)
Affinity DataIC50: 250nMAssay Description:Inhibition of allosterically sensitized mutant form of His6-tagged human HePTP catalytic domain overexpressed in Escherichia coli crude cell lysate u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2020
Entry Details Article
PubMed