Compile Data Set for Download or QSAR
Report error Found 122 Enz. Inhib. hit(s) with all data for entry = 50002074
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453124(CHEMBL4209913)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453125(CHEMBL4214826)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453129(CHEMBL4216242)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453134(CHEMBL4216654)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453139(CHEMBL4205548)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453129(CHEMBL4216242)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453133(CHEMBL4211275)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453126(CHEMBL4208874)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453138(CHEMBL4212209)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453126(CHEMBL4208874)
Affinity DataIC50: 3.90nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453139(CHEMBL4205548)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453137(CHEMBL4217528)
Affinity DataIC50: 4.40nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453125(CHEMBL4214826)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453138(CHEMBL4212209)
Affinity DataIC50: 5.10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)
Affinity DataIC50: 5.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453127(CHEMBL4212762)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453131(CHEMBL4212629)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453124(CHEMBL4209913)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453135(CHEMBL4204975)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453130(CHEMBL4206406)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453130(CHEMBL4206406)
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453128(CHEMBL4207858)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453127(CHEMBL4212762)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453128(CHEMBL4207858)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453130(CHEMBL4206406)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453131(CHEMBL4212629)
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453134(CHEMBL4216654)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453127(CHEMBL4212762)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453127(CHEMBL4212762)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453126(CHEMBL4208874)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453134(CHEMBL4216654)
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453128(CHEMBL4207858)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453131(CHEMBL4212629)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453128(CHEMBL4207858)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453137(CHEMBL4217528)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453133(CHEMBL4211275)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453129(CHEMBL4216242)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453128(CHEMBL4207858)
Affinity DataIC50: 27nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453135(CHEMBL4204975)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50453135(CHEMBL4204975)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
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