Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50002679
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461568(CHEMBL4225198)
Affinity DataKd:  9.40E+3nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461569(CHEMBL4228750)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461570(CHEMBL4224723)
Affinity DataKd: >1.30E+4nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50459942(CHEMBL4227864 | US10730870, Example 85 | US1151208...)
Affinity DataKd:  440nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461570(CHEMBL4224723)
Affinity DataKd:  2.16E+4nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50459942(CHEMBL4227864 | US10730870, Example 85 | US1151208...)
Affinity DataKd:  690nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461568(CHEMBL4225198)
Affinity DataKd:  7.07E+3nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461569(CHEMBL4228750)
Affinity DataKd:  760nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)