Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50002749
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50013727(GW409544 | CHEMBL410478 | CHEBI:79990)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at GAL4-fused human PPARgamma LBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50127222({4-[2-(3-Fluoro-4-trifluoromethyl-phenyl)-4-methyl...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50013727(GW409544 | CHEMBL410478 | CHEBI:79990)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at GAL4-fused human PPARalpha LBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM28706(CHEMBL219586 | 2-methyl-2-{4-[({4-methyl-2-[4-(tri...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  8.90E+3nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  1.83E+4nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462441(CHEMBL1565327)
Affinity DataEC50:  2.50E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in reporter combo cells after 36 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  2.53E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  3.86E+4nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462441(CHEMBL1565327)
Affinity DataEC50:  5.24E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed